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Search Results for " guanfu base a "

4

Compounds

Cat No. Product Name Synonyms Targets
T8182 Guanfu base A Guan-fu base A P450 , Potassium Channel , HER
Guanfu base A is a potent noncompetitive CYP2D6 inhibitor (Ki: 1.20 μM in HLMs; Ki: 0.37 μM for rCYP2D6). It also inhibits HERG channel current.
T8182L Guan-fu base A hydrochloride(1394-48-5 free base) P450
Guan-fu base A hydrochloride is an antiarrhythmic alkaloid was isolated from Aconitum coreanum. Guanfu base A is hydrochloride a CYP2D6 inhibitor of human, monkey, and dog isoforms.
T11510 Guanfu base I Acorine Others
Guanfu base I is an active metabolite of Guanfu base A, isolated from Aconitum coreanum. It have a potent anti-arrhythmic effect.
T11509 Guanfu base H Atisinium chloride Others
Guanfu base H is a diterpenoid alkaloid isolated from Aconitum coreanum. It has antiplasmodial activity against the malarial Plasmodium falciparum strains TM4/8.2 (wild type) and K1CB1 (IC50s: 4 μM and 3.6 μM).
TargetMol